A First-in-Human Study of MEN2312 in Adults With Advanced Breast Cancer

This is a first-in-human study of MEN2312, a lysine acetyltransferase 6 (KAT6) inhibitor, in adult participants with advanced breast cancer.

Trial Details

NCT ID
NCT06638307
Phase
PHASE1
Sponsor
Stemline Therapeutics, Inc.
Status
RECRUITING
Cancer Type
Breast Cancer
Interventions
  • MEN2312
  • Elacestrant
Locations (sample)
  • Springdale, Arkansas, United States|36.18674,-94.12881
  • La Jolla, California, United States|32.84727,-117.2742
  • San Francisco, California, United States|37.77493,-122.41942
  • Santa Monica, California, United States|34.01949,-118.49138
  • New Haven, Connecticut, United States|41.30815,-72.92816

Key Eligibility Criteria

  • Participant has advanced (locoregionally recurrent or metastatic) breast cancer not amenable to curative therapy.
  • Participant must have received at least one prior line of endocrine therapy for advanced/metastatic disease or participant who has radiological evi…
  • Up to 6 prior lines of systemic therapy (including up to 2 prior lines consisting of chemotherapy, cytotoxic antibody drug conjugate, or a combinat…
  • Presence of genetic alterations in PIK3CA/AKT1/PTEN in participants' tumor tissue.

For full eligibility, visit ClinicalTrials.gov.

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